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1

Rifamycins – Obstacles and opportunities

Paul A. Aristoff, George A. Garcia, Paul D. Kirchhoff, H.D. Hollis Showalter

Journal:

Année:

2010

Langue:

english

Fichier:

PDF, 1.09 MB

english, 2010

2

Synthesis and Biological Evaluation of Benzazepine Oxazolidinone Antibacterials.

Paul D. Johnson, Paul A. Aristoff, Gary E. Zurenko, Ronda D. Schaadt, Betty H. Yagi, Charles W. Ford, Judith C. Hamel, Douglas Stapert, Judy K. Moerman

Journal:

Année:

2004

Fichier:

PDF, 148 KB

2004

3

Synthesis of benzopyran prostaglandins, potent stable prostacyclin analogs, via an intramolecular mitsunobu reaction

Paul A. Aristoff, Allen W. Harrison, Anne M. Huber

Journal:

Tetrahedron Letters

Année:

1984

Langue:

english

Fichier:

PDF, 236 KB

english, 1984

4

Synthesis and biological evaluation of benzazepine oxazolidinone antibacterials

Paul D. Johnson, Paul A. Aristoff, Gary E. Zurenko, Ronda D. Schaadt, Betty H. Yagi, Charles W. Ford, Judith C. Hamel, Douglas Stapert, Judy K. Moerman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2003

Langue:

english

Fichier:

PDF, 198 KB

english, 2003

5

Synthesis of binzindene prostaglandins: a novel potent class of stable prostacyclin analogs

Paul A. Aristoff, Allen W. Harrison

Journal:

Tetrahedron Letters

Année:

1982

Langue:

english

Fichier:

PDF, 252 KB

english, 1982

6

Structure-Based Design of Nonpeptidic HIV Protease Inhibitors: The Sulfonamide-Substituted Cyclooctylpyranones

Skulnick, Harvey I., Johnson, Paul D., Aristoff, Paul A., Morris, Jeanette K., Lovasz, Kristine D., Howe, W. Jeffrey, Watenpaugh, Keith D., Janakiraman, Musiri N., Anderson, David J., Reischer, Robert

Journal:

Journal of Medicinal Chemistry

Année:

1997

Langue:

english

Fichier:

PDF, 527 KB

english, 1997

7

Thiadiazolidinones: A new class of alanine racemase inhibitors with antimicrobial activity against methicillin-resistant Staphylococcus aureus

Mihai Ciustea, Sara Mootien, Adriana E. Rosato, Oriana Perez, Pier Cirillo, Kacheong R. Yeung, Michel Ledizet, Michael H. Cynamon, Paul A. Aristoff, Raymond A. Koski, Paul A. Kaplan, Karen G. Anthony

Journal:

Biochemical Pharmacology

Année:

2012

Langue:

english

Fichier:

PDF, 984 KB

english, 2012

8

Total synthesis of a novel antiulcer agent via a modification of the intramolecular Wadsworth-Emmons-Wittig reaction

Aristoff, Paul A., Johnson, Paul D., Harrison, Allen W.

Journal:

Journal of the American Chemical Society

Année:

1985

Langue:

english

Fichier:

PDF, 1.10 MB

english, 1985

9

Tipranavir (PNU-140690): A Potent, Orally Bioavailable Nonpeptidic HIV Protease Inhibitor of the 5,6-Dihydro-4-hydroxy-2-pyrone Sulfonamide Class∇

Turner, Steve R., Strohbach, Joseph W., Tommasi, Ruben A., Aristoff, Paul A., Johnson, Paul D., Skulnick, Harvey I., Dolak, Lester A., Seest, Eric P., Tomich, Paul K., Bohanon, Michael J.

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 322 KB

english, 1998

10

Reaction of CC-1065 and select synthetic analogs with DNA

Laurence H. Hurley, Chong-Soon Lee, J.Patrick McGovren, Martha A. Warpehoski, Mark A. Mitchell, Robert C. Kelly, Paul A. Aristoff

Journal:

Biochemical Pharmacology

Année:

1988

Langue:

english

Fichier:

PDF, 176 KB

english, 1988

11

Kinetic studies with the non-nucleoside human immunodeficiency virus type-1 reverse transcriptase inhibitor U-90152E

Irene W. Althaus, James J. Chou, Andrea J. Gonzales, Martin R. Deibel, Chou Kuo-Chen, Ferenc J. Kezdy, Donna L. Romero, Richard C. Thomas, Paul A. Aristoff, W.Gary Tarpley, Fritz Reusser

Journal:

Biochemical Pharmacology

Année:

1994

Langue:

english

Fichier:

PDF, 1.40 MB

english, 1994

12

Oxazolidinones: a new class of antibacterials

Gary E Zurenko, John K Gibson, Dean L Shinabarger, Paul A Aristoff, Charles W Ford, W.Gary Tarpley

Journal:

Current Opinion in Pharmacology

Année:

2001

Langue:

english

Fichier:

PDF, 155 KB

english, 2001

13

Antibody-Drug Conjugates for the Treatment of Cancer

Flygare, John A., Pillow, Thomas H., Aristoff, Paul

Journal:

Chemical Biology & Drug Design

Année:

2013

Langue:

english

Fichier:

PDF, 848 KB

english, 2013

14

Structure-Based Design of HIV Protease Inhibitors: Sulfonamide-Containing 5,6-Dihydro-4-hydroxy-2-pyrones as Non-Peptidic Inhibitors ¶

Thaisrivongs, Suvit, Skulnick, Harvey I., Turner, Steve R., Strohbach, Joseph W., Tommasi, Ruben A., Johnson, Paul D., Aristoff, Paul A., Judge, Thomas M., Gammill, Ronald B., Morris, Jeanette K., Rom

Journal:

Journal of Medicinal Chemistry

Année:

1996

Langue:

english

Fichier:

PDF, 184 KB

english, 1996

15

PRACTICAL SYNTHESIS OF 3,3,4,4-TETRAMETHYLCYCLOPENTANONE

Aristoff, Paul A., Nelson, Cynthia L.

Journal:

Organic Preparations and Procedures International

Année:

1983

Langue:

english

Fichier:

PDF, 194 KB

english, 1983

16

Structure-Based Design of HIV Protease Inhibitors: 5,6-Dihydro-4-hydroxy-2-pyrones as Effective, Nonpeptidic Inhibitors

Thaisrivongs, Suvit, Romero, Donna L., Tommasi, Ruben A., Janakiraman, Musiri N., Strohbach, Joseph W., Turner, Steve R., Biles, Carolyn, Morge, Raymond R., Johnson, Paul D., Aristoff, Paul A., Tomich

Journal:

Journal of Medicinal Chemistry

Année:

1996

Langue:

english

Fichier:

PDF, 1.11 MB

english, 1996

17

Inhibition of mycobacterial alanine racemase activity and growth by thiadiazolidinones

Lee, Yashang, Mootien, Sara, Shoen, Carolyn, Destefano, Michelle, Cirillo, Pier, Asojo, Oluwatoyin A., Yeung, Kacheong R., Ledizet, Michel, Cynamon, Michael H., Aristoff, Paul A., Koski, Raymond A., K

Journal:

Biochemical Pharmacology

Année:

2013

Langue:

english

Fichier:

PDF, 1.74 MB

english, 2013

18

Benzindene prostaglandins. Synthesis of optically pure 15-deoxy-U-68,215 and its enantiomer via a modified intramolecular Wadsworth-Emmons-Wittig reaction

Lin, Chiu Hong, Aristoff, Paul A., Johnson, Paul D., McGrath, James P., Timko, Joseph M., Robert, Andre

Journal:

Journal of Organic Chemistry

Année:

1987

Langue:

english

Fichier:

PDF, 1.15 MB

english, 1987

19

Experiments directed toward the total synthesis of terpenes. 23. Synthesis of 4a-methyl-4,4a,7,8-tetrahydro-9H-benzocycloheptene-2(3H),5(6H)-dione (B-homo Wieland-Miescher ketone): a versatile intermediate for terpene synthesis

Ireland, Robert E., Aristoff, Paul A., Hoyng, Charles F.

Journal:

Journal of Organic Chemistry

Année:

1979

Langue:

english

Fichier:

PDF, 761 KB

english, 1979

20

Molecular basis for sequence-specific DNA alkylation by CC-1065

Hurley, Laurence H., Lee, Chong Soon, McGovren, J. Patrick, Warpehoski, Martha A., Mitchell, Mark A., Kelly, Robert C., Aristoff, Paul A.

Journal:

Année:

1988

Langue:

english

Fichier:

PDF, 2.32 MB

english, 1988

21

Sequence-selective guanine reactivity by duocarmycin A

Mitchell, Mark A., Weiland, Katherine L., Aristoff, Paul A., Johnson, Paul D., Dooley, Thomas P.

Journal:

Chemical Research in Toxicology

Année:

1993

Langue:

english

Fichier:

PDF, 1.67 MB

english, 1993

22

Antibacterial Oxazolidinones Possessing a Novel C-5 Side Chain. (5 R )- trans -3-[3-Fluoro-4- (1-oxotetrahydrothiopyran-4-yl)phenyl]-2- oxooxazolidine-5-carboxylic Acid Amide (PF-00422602), a New Lead Compound

Poel, Toni-Jo, Thomas, Richard C., Adams, Wade J., Aristoff, Paul A., Barbachyn, Michael R., Boyer, Frederick E., Brieland, Joan, Brideau, Roger, Brodfuehrer, Joanne, Brown, Alan P., Choy, Allison L.,

Journal:

Journal of Medicinal Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 57 KB

english, 2007

23

Coupling of cyclopropapyrroloindole (CPI) derivatives. The preparation of CC-1065, ent-CC-1065, and analogs

Kelly, Robert C., Gebhard, Ilse, Wicnienski, Nancy, Aristoff, Paul A., Johnson, Paul D., Martin, David G.

Journal:

Journal of the American Chemical Society

Année:

1987

Langue:

english

Fichier:

PDF, 270 KB

english, 1987

24

Synthesis of 9-substituted carbacyclin analogs

Aristoff, Paul A., Johnson, Paul D., Harrison, Allen W.

Journal:

Journal of Organic Chemistry

Année:

1983

Langue:

english

Fichier:

PDF, 1.08 MB

english, 1983

25

Experiments directed toward the total synthesis of terpenes. 24. On the .pi. route to aphidicolin: synthesis of 18,19-bisnoraphidicolan-3-one

Ireland, Robert E., Aristoff, Paul A.

Journal:

Journal of Organic Chemistry

Année:

1979

Langue:

english

Fichier:

PDF, 1.33 MB

english, 1979

26

Practical synthesis of 6a-carbaprostaglandin I2

Aristoff, Paul A.

Journal:

Journal of Organic Chemistry

Année:

1981

Langue:

english

Fichier:

PDF, 652 KB

english, 1981

27

Improved method for the conversion of enol lactones to cyclic .alpha.,.beta.-unsaturated ketones

Aristoff, Paul A.

Journal:

Journal of Organic Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 290 KB

english, 1985

28

Synthesis and biochemical evaluation of the CBI-PDE-I-dimer, a benzannelated analog of (+)-CC-1065 that also produces delayed toxicity in mice

Aristoff, Paul A., Johnson, Paul D., Sun, Daekyu, Hurley, Laurence H.

Journal:

Journal of Medicinal Chemistry

Année:

1993

Langue:

english

Fichier:

PDF, 3.79 MB

english, 1993

29

Reductive aromatization of quinols. New convenient methods for the regiospecific synthesis of p-hydroxy C-aryl glycals

Parker, Kathlyn A., Coburn, Craig A., Johnson, Paul D., Aristoff, Paul

Journal:

Journal of Organic Chemistry

Année:

1992

Langue:

english

Fichier:

PDF, 541 KB

english, 1992

30

Interstrand DNA cross-linking with dimers of the spirocyclopropyl alkylating moiety of CC-1065

Mitchell, Mark A., Johnson, Paul D., Williams, Marta G., Aristoff, Paul A.

Journal:

Journal of the American Chemical Society

Année:

1989

Langue:

english

Fichier:

PDF, 836 KB

english, 1989

31

Synthesis of CBI-PDE-I-dimer, the benzannelated analog of CC-1065

Aristoff, Paul A., Johnson, Paul D.

Journal:

Journal of Organic Chemistry

Année:

1992

Langue:

english

Fichier:

PDF, 934 KB

english, 1992

32

General procedure for the synthesis of o-aminophenylacetates by a modification of the Gassman reaction

Johnson, Paul D., Aristoff, Paul A.

Journal:

Journal of Organic Chemistry

Année:

1990

Langue:

english

Fichier:

PDF, 292 KB

english, 1990

33

A Novel Riboswitch-Binding Flavin Analog that Protects Mice Against Clostridium difficile Infection without Inhibiting Cecal Flora

Blount, Kenneth F., Megyola, Cynthia, Plummer, Mark, Osterman, David, O'Connell, Tim, Aristoff, Paul, Quinn, Cheryl, Chrusciel, R. Alan, Poel, Toni J., Schostarez, Heinrich J., Stewart, Catherine A, W

Journal:

Antimicrobial Agents and Chemotherapy

Année:

2015

Langue:

english

Fichier:

PDF, 961 KB

english, 2015

34

On the Stereochemistry of E′- and E′-Reactions

Vogel, Ernst, Caravatti, Giorgio, Franck, Peter, Aristoff, Paul, Moody, Christopher, Becker, Anna-Maria, Felix, Dorothee, Eschenmoser, Albert

Journal:

Chemistry Letters

Année:

1987

Langue:

english

Fichier:

PDF, 8.19 MB

english, 1987

35

New Classes of Alanine Racemase Inhibitors Identified by High-Throughput Screening Show Antimicrobial Activity against Mycobacterium tuberculosis

Anthony, Karen G., Strych, Ulrich, Yeung, Kacheong R., Shoen, Carolyn S., Perez, Oriana, Krause, Kurt L., Cynamon, Michael H., Aristoff, Paul A., Koski, Raymond A., Ahmed, Niyaz

Journal:

Année:

2011

Langue:

english

Fichier:

PDF, 635 KB

english, 2011

36

Structure-activity relationship of flavin analogs that target the FMN riboswitch

Vicens, Quentin, Mondragón, Estefanía, Reyes, Francis E., Coish, Philip, Aristoff, Paul, Berman, Judd, Kaur, Harpreet, Kells, Kevin W., Wickens, Phil, Wilson, Jeffrey, Gadwood, Robert C., Schostarez,

Journal:

ACS Chemical Biology

Année:

2018

Langue:

english

Fichier:

PDF, 2.00 MB

english, 2018